ZheJiang Holypharm Blotech Co.,Ltd.
Pharma Division          
Veterinary Division     
Agrochemical Division
Hot Products          
Developing Products          

Marketing list

Cardiovascular & its advanced intermediates
 (including R&D products)

Atorvastatin & ATS-5 ATS-8 ATS -9 M 4 L 1
ATS-5 : (R)-4-cyano-3-hydroxybutyric acid ethyl ester
ATS-8 : (4R,Cis)-1,1-dimethylethyl-cyanomethyl-2,2- dimethyl-1,3-dioxane-4-acetate

CAS NO.: 134523-00-5
CAS NO.: 141942-85-0
CAS NO.: 125971-94-0

Fluvastatin & F2,F4
F4 : Tert- butyl( E)-3,5-dihydroxy-7-[3'-(4"-fluorophenyl)-1'- methylethyl-indol-2'-yl] hept-6-enoate

CAS N O .: 59333-67-4

Rosuvastatin Calcium & Z7,Z8,R3
Z-7 : 4-(4- Fluorophenyl)-6-isopropyl-2-[ (N- methyl-N-methylsulfonyl)amino]pyrimidine-5-yl-methonol

CAS No.: 147098-20-2
CAS No.: 147118-36-3

 

Ramipril & intermediate
(1S, 3S, 5S)-2-azabicyclo [3,3,0] octane-3-carborylic acid benzyl ester hydrochloride

CAS No.: 87333-19-5

Lisinopril
N2-[(1S)-ethoxycarbonyl-3-phenylpropyl]-N6-Trifluoroacetyl-L-Lysine

CAS No.: 83915-83-7
CAS No: 116169-90-5

Enalapril
N2-[(S)-(+)-1-(Ethoxy carbonyl)-3-phenylpropyl]-L-Alanine ECPPA

CAS No.: 76095-16-4
CAS No.: 82717-96-2

Benazepril
T ert-butyl-(s)-(3-amino-2-oxo-2,3,4,5-tetrahydobenzo[b]azepine-1yl) Acetate

CAS No.: 86541-74-4
CAS No.: 109010-60-8

Perindopril
(2S,3As,7As)-octahydroindole-2-carboxylic acid
N-[(S)-1-carbethoxybutyl]-(S)-alanine

CAS No.: 82834-16-0
CAS No. 80875-98-5
CAS No. 8 2834-12-6

Quinapril
S-1,2,3,4 ¨C tetrahydro-3-isoquinolinecarboxylic acid

CAS No.: 85441-61-8

 

Valsartan
N-[[(2-cyano(1.1-biphenyl)-4-yl)methyl]methyl ester]-L- valine.hydrochloride

CAS No.: 137862-53-4

Telmisartan & Int.
4-[ 2'-n-propyl-1, 4'-dimethyl-(2,6-dibenzimidazole)-1'-yl] methylene (1, 1'-biphenyl)-2-methyl formate

CAS No.: 144701-48-4
CAS No.: 144702-26-1

Candesartan Cilexetil
N-( Triphenylmethyl) ¨C 5-( 4'-bromomethylbiphenyl-2yl) tetrazole

CAS No.: 145040-37-5
CAS No.: 124750-51-2

Losartan Potassium
N-(Triphenylmethyl)-5-(4'-Bromomethylbiphenyl-2-Yl-) Tetrazole
2-N-butyl-4-(5,5)-chloro-5-hydroxymethanol imidazole

CAS No.: 12475-99-8
CAS No.: 124750-51-2

Olmesartan & int
4-chloromethyl-5-methyl-1,3-Dioxol-2-one (DMDO-CL)

 CAS NO: 144689-63-4
 CAS No.: 80841-78-7

Irbesartan
2n-Butyl-4(5)-chloro-1H-Imidazole-5(4)-Oarboxaldehyde

CAS No.: 13 8402-11-6
CAS No.: 83857-96-9

Doxazosin
 N-(1,4-Benzodioxan-2-Yl-Carbonyl)Piperazine

CAS No.: 77883-43-3
CAS No.: 70918-00-2

Clopidogrel
2-Thiophene Ethanol
(+)-Methyl-alpha-(2-Thienylethamino) (2-Chlorophenyl) AcetateHydrochloride
N-[(2-Thienyl)ethyl]-(2s)-2-chloro-phenyl Glycine methyl ester

CAS No.: 113665-84-2
CAS No.: 5402-55-1
CAS No.: 141109-19-5
CAS No.: 5680-79-5

Cilostazole
5-(4-Chlorobutyl)-1-Cyclohexyl-1H-Tetrazole
6-Hydroxy-3,4-dihydro-2(1H)-quinolinone

CAS No.: 73963-72-1
 CAS No.: 73963-42-5
CAS No.: 54197-66-9

Cilnidipine
Methylethyl-3-Nitro Benzylidene Acetoacetate

CAS NO: 132203-70-4

Loratadine & int

 

Carvedilol & int
4-Hydroxy-9H-carbazole
Epoxy propoxy carbazol

CAS No : 7 2956-09-3
CAS No.: 54989-33-2

Cilostazole
5-(4-Chlorobutyl)-1-Cyclohexyl-1H-Tetrazole
6-Hydroxy-3,4-dihydro-2(1H)-quinolinone

CAS No.: 73963-72-1
CAS No.: 73963-42-5
CAS No.: 54197-66-9

Ezitimibe & int
(s)-4-phenyl-2-Oxazolidione
3-[5-(4-fluorophenyl)-1,5-dioxopentyl]-4-phenyl-(4S)-2-oxazolidinone

CAS NO: 163222-33-1
CAS No.: 99395-88-7
189028-93-1

Anti- cancer & its advanced intermediates
(including R&D products)

Gemcitabine &int
2-Deoxy-2,2-difluoro-D-ribofuranose-3,5-dibenzoate
2-Deoxy-2,2-difluoro-D-ribofuranose-3,5-di benzoate-1-methane sulfonate

CAS N o : 95058-81-4

CAS No: 143157-22-6

Bicalutamide &int
4-cyano-3-trifluoro methyl aniline
4-Fluorothiophenol
N-[4-Cyano-3-(trifluoromethyl)phenyl]-3-[(4-fluorophenyl)thio]-2-hydroxy-2-methylpropionamide

CAS No.: 9 0357-06-5


CAS No.: 90356-78-8

Anastrazole & int
2-[3-(Cyano-dimethyl-methyl)-5-methyl-phenyl]-2-methyl-propionitrile

CAS N o .:120511-73-1
CAS N o .: 120511-72-0

Granisetron & int

 

Palonosetron HCl & int
S-(-)-3-Aminoquinuclidine 2HCl
N-(1-azabicyalo[2,2,2]oct-3S-yl)-1,2,3,4-tetrahydronaphthalen-1S-ylcarboxamine


119904-90-4

Bisoprolol & int

 

Letrozole & int
4-[a-(4-cyanophenyl)-chloromethyl]-benzonitrile

112809-51-5
112809-57-1

Ibandronate Sodium
3-(N-methylpentylamino)propionic acid hydrochloride

 

Anti-depressant & its advanced intermediates
(including R&D products)

Rivastigmine
N-Ethyl-N-Methylcarbamoyl Chloride

CAS NO: 12 3441-03-2
CAS No.: 42252-34-6

Aripiprazole
3,4-dihydro-7-Hydroxy-2(1H)-Quinolinone
N-(2,3-dichlorophenyl) Piperazine Hydrochloride

CAS NO: 12 9722-12-9
CAS NO.: 22246-18-0
CAS NO.: 41202-77-1

Carbamazepine

 

Oxcarbazepine

 

Sumatriptan Succinate
N-Methyl-4-Nitro Benzene Methane Sulfonamide
4-Hydrazine phenyl ¨C N-methyl methane sulfonamide

 CAS No.: 103628-46-2

Naratriptan
2-(1-Methyl-4-Piperidinyl)-Acetaldehyde
N-Methyl-1H-Indole-5-Ethane Sulfonamide
N-Methyl-4-Piperidinol

CAS NO: 121679-13-8


CAS No. 106-52-5

Zolmitriptan
 (S)-4-(4-Aminobenzyl)-2-Oxazolidinone
4-nitro-L-phenylalanino

CAS NO: 139264-17-8
CAS No. 152305-23-2
CAS No. 949-99-5

Donepezil
 5,6-Dimethoxy-1-Indanone
N-Benzyl Piperidine-4-Carboxaldehyde

CAS No.: 12 0014-06-4
CAS No.: 2107-69-9

Rizatriptan
4-(1H-1,2,4-Triazole-1-Yl Methyl) Aniline Hcl

CAS NO: 145202-66-0

Ciclopirox Olamine

CAS NO: 29342-05-0

Venlafaxine
2-(1-Hydroxy Cyclohexyl)-2-(4-Methoxy Phenyl) Acetonitrile

CAS NO: 99300-78-4

Risperidone
3-(2-Chloroethyl)-6,7,8,9-Tetrahydro-2-Methyl-4H-Pyridin [1,2-a]-pyrimidine ¨C4-one
6-Fluoro-3-(4-piperidinyl) ¨C 1,2-benzisoxazole

CAS NO: 10 6266-06-2
CAS No.: 41078-70-0
CAS No.: 84163-77-9

Ziprasidone
5-Chloroacetyl-6-Chloro-1,3-Dihydro-2-H Indole-2-One

CAS No.: 138982-67-9

Levetiracetam

 

Paroxetine

CAS NO: 6 1869-08-7

Duloxetine
(S)-N,N-dimethyl-gamma-(1-naphthalenyloxy)-2-thiophenepropanamine oxalate

CAS NO: 136434-34-9

Gabapentin & int CDA CAM
1,1-Cyclohexane Diacetic Acid Monoamide ( CAM )
1,1-Cyclohexane Diacetic Anhydride( CAA )

CAS NO: 60142-96-3
CAS No: 99189-60-3

Pregabalin

CAS No: 148553-50-8

Tegaserod
N-Amino-N-Pentylguanidine Hydroiodide

 CAS NO: 189188-57-6

olanzapine
4-Amino-2-Methyl-10H-Thieno[2,3-b][1,5]Benxodiazepine Hcl

CAS NO: 132539-06-1
CAS No. 138564-60-0

Clozapine

 

ZOPICLONE
6-(5-chloropyrid-2yl)-5-hydroxy-7oxo-5,6-dihydro-pyrrolo-(3,4b)-pyrazine

CAS NO : 43200-80-2

Topiramate

 

anti-diabetes drug & its advanced intermediates
 (including R&D products)

Acarbose

CAS NO: 56180-94-0

Voglibose
Valiolamine

CAS NO: 83480-29-9

Tamsulosin
R-(-)-5-(2-Amino-propyl)-2-methoxy-benzenesulfonamide
2-(2-Ethoxyphenoxy)bromide ethane

CAS NO: 106133-20-4
CAS No. 112101-81-2
CAS No. 3259-03-8

 

glimepiride   

 

Repaglinide

 

Rimonabant

 

Miglitol

 

steroid drug & its advanced intermediates
 (including R&D products)

Cyproterone Acetate
1, 2a -Methylene-6-didehydro -17a -acetoxy Progesterone
1-Chloromethyl-6-chloro-6-dehydro -17a -acetoxy Progesterone

CAS:427-51-0

Mifepristone

CAS: 84371-65-3

Finasteride

CAS: 98319-26-7

Eplerenone
11alpha-Hydroxy canrenone

CAS: 107724-20-9
CAS:192569-17-8

Methylprednisolone

CAS:83-43-2

Fluticasone propionate

CAS: 80474-14-2

Conjugated Estrogens

 

Exemestane

CAS: 107868-30-4

Fluoxymesterone

CAS: 76-43-7

Fluorogestone acetate

CAS: 337-03-1

Budesonide
16-Alpha-Hydroxy Prednisolone

CAS: 51333-22-3

Drospirenon

CAS: 67392-87-4

Triamcinolone Acetonide

CAS: 76-25-5

Megestrol Acetate

CAS:595-33-5

Deflazacort

CAS: 14484-47-0

Estrone

CAS: 53-16-7

Dydrogesterone

CAS: 152-62-5

Medrogestone

CAS: 977-79-7

Fluocinolone Acetonide

CAS:67-73-2

Hydrocortisone

CAS: 50-23-7

Hydrocortisone Acetate

CAS: 50-03-3

Antibiotics and their intermediates
(Including R&D products)

SMIA
Sin-Methoxyimino Furanyl Acetic Acid Ammonium Salt

97148-89-5

EHATA
Ethyl(Z)-2-(2-Aminothiazole-4-yl)-2-Methoxyimino Acetate

64485-88-7

TAA
1,2,3,4-Tetrazolyl-1- Acetic Acid

21732-17-2

MMT
5-Mercapto-1-methyl tetrazole

13183-79-4

MMTA
2-(2-Mercapto-4-Methyl-1,3-Thiazole-5-yl) Acetic Acid

34272-64-5

MICA ACID
(Z)-2-(tert-methoxycarbonyl methoxyimino)-2-(2-aminothiazol-4-yl) acetic acid

80554-17-8

MICA ESTER
S-2-benzothiazolyl (Z)-2-(2-aminothiazol-4-yl)-2-methoxycarbonylmethoxyiminothio acetate

246035-38-1

MAEM
2-Mercaptobenzothiazoyl (Z)-2-(2-Aminothiazole-4-yl)-2-methoxyimino acetate

80756-85-0

TTZ
1,2,5,6-Tetrahydro-2-methyl-5,6-dioxo-1,2,4-triazine

58909-39-0

HO-EPCP
a -{[(4-Ethyl-2,3-Dioxo-1-Piperazinyl)Carbonyl] Amino}-4-Hydroxy-Benzene Acetic Acid

62893-24-7

CPP
2,3-cyclopenteno pyridine

533-37-9

CHP
2,3-cyclohexano pyridine

10500-57-9

Ofloxacin
Olfoxacin Acid

82419-36-1
82419-35-0

Levofloxacin
Levofloxacin Acid
2,3,4,5-tetrafluoro benzoic acid

100986-85-4
100986-89-8
1201-31-6

Gatifloxacin

180200-66-2

Ciprofloxacin Hcl
Q-acid

86393-32-0
86393-33-1

 

Aciclovir

59277-89-3

Famciclovir

104227-87-4

Ganciclovir

82410-32-0

Valaciclovir

124832-26-4

Meropenem & 4-AA 4-BMA MAP

 

Penipenem 4-nitrobenzyl-1-((S)-3-mercaptopyrrolidin-1-yl)ethylidenecarbamate

 

Farop enem & int

 122547-49-3

Biapenem
6,7-dihydro-6-mercapto-5H-pyrazolo[1,2-a][1,2,4]triazolium chloride or
6,7-dihydro-6-mercapto-5H-pyrazolo[1,2-a][1,2,4]triazol-4-ium,chloride

120410-24-4

153851-71-9

Ertapenem

 

Imipenem

74431-23-5

1H-1,2,3-Triazole

288-36-8

Tetramethyl Guanidine

80-70-6

Clarithromycin

8 1103-11-9

Azitromycin

8 3905-01-5

Amorolfine

106614-68-0

Terbinafine

78628-80-5

Ciclopirox Olamine

29342-05-0

Other item and their intermediates
(Including R&D products)

Isotretinoin

 

Iohexol

 

Sucralose

 

Co enzyme Q10

 

Doxofylline

 

Calcipotriol

 

Glucosamine Sulfate K + ; Na + ; HCL

 

Efavirienz Int. : Cyclopropyl acetylene
                     Cyclopropyl methylketone
                     2-trifluoroacetyl ¨C4-chlorophenylamine HCL

 

Abacavir

 

Amorolfine

 

Atovaquone

 

Donepezil

 

Diethylstilbestrol

 

Etodolac

 

Modafinil

 

Montelucastan

 

Sildenafil Citrate

 

Valaciclovir Hcl

 

Verapamil

 

Moxifloxacin

 

R&D list

Naratriptan

2-(1-Methyl-4-Piperidinyl)-Acetaldehyde
N-Methyl-1H-Indole-5-Ethane Sulfonamide
N-Methyl-4-Piperidinol

Rivastigmine

N-Ethyl-N-Methyl carbamoyl Chloride
Di-P-Tolyl Tartaric Acid
Palonosetron
Bicalutamide

 

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